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NF-56-EJ40 hydrochloride
CAS No. 2728500-80-7
NF-56-EJ40 hydrochloride( —— )
Catalog No. M33038 CAS No. 2728500-80-7
NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 48 | Get Quote |
|
| 10MG | 71 | Get Quote |
|
| 25MG | 118 | Get Quote |
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| 50MG | 177 | Get Quote |
|
| 100MG | 258 | Get Quote |
|
| 200MG | 388 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameNF-56-EJ40 hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionNF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1.
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DescriptionNF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 hydrochloride has high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetGHSR
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RecptorGHSR
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Research Area——
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Indication——
Chemical Information
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CAS Number2728500-80-7
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Formula Weight516.46
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Molecular FormulaC27H31Cl2N3O3
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(CC1=C(NC(C2=CC=CC(C3=CC=C(CN4CCN(CC4)C)C=C3)=C2)=O)C=CC=C1)O.Cl.Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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